Seznam steroidních antiandrogenů - List of steroidal antiandrogens

Cyproteron-acetát, nejznámější a nejpoužívanější steroidní antiandrogen.

Steroid kruhový systém.

Tohle je seznam steroidní antiandrogeny.

Deriváty progesteronu

• 11α-hydroxyprogesteron = 11α-hydroxyprogesteron
• Chlormadinonacetát = 17a-acetoxy-6-chlor-5⁶-progesteron
• Klometeron (L-38000) = 6a-chlor-16a-methylprogesteron
• Cyproteron (SH-80881) = 1,2a-methylen-6-chlor-5⁶-17a-hydroxyprogesteron
• Cyproteron-acetát = 1,2α-methylen-6-chlor-5⁶-17a-acetoxyprogesteron
• Edogestron (PH-218) = 17a-acetoxy-3,3-ethylendioxy-6-methylpregn-5-en-20-on
• Medrogeston = 6,17a-dimethyl-8⁶-progesteron
• Megestrol-acetát = 17a-acetoxy-5⁶-6-methylprogesteron
• Nomegestrol-acetát = 17a-acetoxy-5⁶-6-methyl-19-norprogesteron
• Osateronacetát (TZP-4238) = 17a-acetoxy-6-chlor-2-oxa-5⁶-progesteron

Deriváty testosteronu

• Abirateron (CB-7598) = 17- (3-pyridinyl) androsta-5,16-dien-3β-ol
• Abirateronacetát = 17- (3-pyridinyl) androsta-5,16-dien-3p-ol-acetát
• Benorterone (SKF-7690, FC-612) = 17α-methyl-B-nortestosteron
• BOMT (Ro 7-2340) = 6α-brom-4-oxa-17α-methyl-4,5α-dihydrotestosteron
• Delanteron (GBR-21162) = 17p-dehydroxy-la-methyl-5¹⁶-testosteron
• Dienogest = 17a-kyanomethyl-19-nor-5⁹⁽¹⁰⁾-testosteron
• Epitestosteron = 17α-epitestosteron
• Galeterone (TOK-001, VN / 124-1) = 17- (lH-benzimidazol-l-yl) androsta-5,16-dien-3p-ol
• Metogest (SC-14207) = 16,16-dimethyl-19-nortestosteron
• Mifepriston = Llp- [p- (dimethylamino) fenyl] -17- (l-propinyl) -5⁹-19-nortestosteron
• Oxendolon (TSAA-291) = 16p-ethyl-19-nortestosteron
• Rosterolon (SH-434, 17α-propylmesterolon) = 1α-methyl-17α-propyl-4,5α-dihydrotestosteron
• Topteron (WIN-17665) = 17α-propyltestosteron
• Trimethyltrienolon (R-2956, RU-2956) = 2α, 2β, 17α-trimethyl-19-nor-δ^9,11-testosteron
• Zanoteron (WIN-49596) = (5a, 17a) -l '- (methylsulfonyl) -l'-H-pregn-20-ino [3,2-c] pyrazol-17-ol

Spirolaktonové deriváty

• SC-5233 (spirolakton) = 17α- (2-karboxyethyl) testosteron γ-lakton
• SC-8109 = 19-norspirolakton
• Canrenone (aldadien) = A⁶-spirolakton
• Dicirenon (SC-26304) = 7a-karboxyisopropylspirolakton
• Drospirenon = 6p, 7p: 15p, 16p-dimethylenespirolakton
• Mespirenon (ZK-94679) = Δ¹-7a-acetylthio-15p, 16p-methylenespirolakton
• Mexrenone (ZK-32055, SC-25152) = 7α- (methoxykarbonyl) spirolakton
• Prorenon (SC-23133) = 6a, 7a-methylenespirolakton
• Spironolakton = 7α-acetylthiospirolakton
• Spirorenon (ZK-35973) = Δ¹-6p, 7p: 15p, 16p-dimethylenespirolakton
• Spiroxason = 7α-acetylthiospirolakton s odstraněním ketonové skupiny z C17α spirolaktonového kruhu

Deriváty kortizolu

• 9,11-dehydrocortexolon 17a-butyrát (CB-03-04) = 17α- (butyryloxy) -9,11-didehydrodeoxykortikosteron
• Clascoteron (CB-03-01; cortexolon 17α-propionát, 11-deoxykortizol 17α-propionát) = 17α- (propionyloxy) deoxykortikosteron

Ostatní

• Guggulsteron = pregna-4,17-dien-3,16-dion
• Nordinone = 11α-hydroxy-17,17-dimethyl-18-norandrosta-4,13-dien-3-on

Viz také

• Seznam steroidů